Each 5 mg film-coated tablet contains 8.078 mg of tofacitinib citrate equivalent to 5 mg of tofacitinib free base active pharmaceutical ingredient. Each 5 mg tablet also contains 61.307 mg lactose monohydrate.
Excipients/Inactive Ingredients: Microcrystalline cellulose, Lactose monohydrate, Croscarmellose sodium, Magnesium stearate.
Film Coat for 5 mg tablets: Opadry II White (33G28523) containing: HPMC 2910/Hypromellose 6cP, Titanium dioxide, Lactose monohydrate, Macrogol/PEG3350, Triacetin (glycerol triacetate).