Rexulti

Rexulti Drug Interactions

brexpiprazole

Manufacturer:

Otsuka (Philippines)

Distributor:

Otsuka (Philippines)
Full Prescribing Info
Drug Interactions
Drugs Having Clinically Important Interactions with Brexpiprazole (Rexulti): See Table 12.

Click on icon to see table/diagram/image

Drugs Having No Clinically Important Interactions with Brexpiprazole (Rexulti): Based on pharmacokinetic studies, no dosage adjustment of Brexpiprazole (Rexulti) is required when administered concomitantly with CYP2B6 inhibitors (e.g., ticlopidine) or gastric pH modifiers (e.g., omeprazole). Additionally, no dosage adjustment for substrates of CYP2D6 (e.g., dextromethorphan), CYP3A4 (e.g., lovastatin), CYP2B6 (e.g., bupropion), BCRP (e.g., rosuvastatin), or P-gp (e.g., fexofenadine) is required when administered concomitantly with Brexpiprazole (Rexulti).
Register or sign in to continue
Asia's one-stop resource for medical news, clinical reference and education
Already a member? Sign in
Register or sign in to continue
Asia's one-stop resource for medical news, clinical reference and education
Already a member? Sign in