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Each tablet contains: Baclofen 10 mg.
Baclofen is an effective muscle relaxant and antispastic agent with a spinal site of action. Baclofen is structurally similar to the inhibitory neurotransmitter gamma-amino-butyric acid, though its actions are different. It is stereospecifically to GABAB receptors. It is thought that activation of the GABAB receptors on presynaptic terminal reduces evoked transmitter release, perhaps through reduced presynaptic Ca2+ influx. Baclofen can inhibit the function of inward calcium currents in some cells. The drug rapidly absorbed after oral administration and is widely distributed throughout the body.
