Zifagra

Zifagra

sildenafil

Manufacturer:

Ifars
Concise Prescribing Info
Contents
Sildenafil
Indications/Uses
Erectile dysfunction.
Dosage/Direction for Use
50 mg an hr prior to sexual activity. Max: 100 mg once daily. May be reduced to 25 mg.
Contraindications
Hypersensitivity.
Special Precautions
Antacid may be given in ½ hr interval. Patients w/ CV disease, non-arteritic anterior ischemic optic neuropathy (NAION), visual impairment or loss; hypotension at rest (BP <90/50 mmHg) or HTN at rest (BP 170/110 mmHg); heart failure or CAD causing unstable angina; retinitis pigmentosa. Patients who have suffered from MI, stroke, or life-threatening arrhythmias in the past 6 mth. Prolonged erection of >4 hr & priapism (painful erection of >6 hr). Patient w/ renal failure & dialysis. Pregnancy & lactation. Childn.
Adverse Reactions
Facial edema, photosensitivity reactions, shock, asthenia, pain, chills, accidental falls, abdominal pain, allergic reactions, chest pain, accidental injury; CV disorders; vomiting, glossitis, colitis, dysphagia, gastritis, gastroenteritis, esophagitis, stomatitis, dry mouth, abnormal LFTs, rectal bleeding, gingivitis; anemia & leukopenia; unstable sugar levels, hyperglycemia, peripheral edema, hyperuricemia, hypoglycemic reactions, hypernatremia; musculoskeletal arthritis, arthrosis, myalgia, muscle tears, tenosynovitis, bone pain, myasthenia, synovitis; ataxia, hypertonia, neuralgia, neuropathy, paraesthesia, tremor, vertigo, depression, insomnia, somnolence, abnormal dreams, decreased reflexes, hypesthesia; asthma, dyspnea, laryngitis, pharyngitis, sinusitis, bronchitis, increased sputum, increased cough frequency; urticaria, herpes simplex, pruritus, sweating, skin wounds, contact dermatitis, exfoliative dermatitis; mydriasis, conjunctivitis, photophobia, tinnitus, eye pain, deafness, ear pain, bleeding in the eyes, cataracts; cystitis, nocturia, urinary frequency, breast enlargement, urinary incontinence, abnormal ejaculation, genital edema & anorgasmia.
Drug Interactions
Reduced clearance w/ CYP3A4 (eg, ketoconazole, erythromycin, cimetidine) or CYP2C9 inhibitors. Increased clearance w/ CYP3A4/2C9 inducers. Increased plasma conc w/ cimetidine. Increased AUC w/ erythromycin. Increased Cmax & AUC w/ saquinavir, ritonavir. Decreased AUC & Cmax w/ bosentan. Increased AUC & Cmax of bosentan. Decreased plasma level w/ rifampin. May lead to symptomatic hypotension w/ α-blocker.
MIMS Class
Drugs for Erectile Dysfunction & Ejaculatory Disorders
ATC Classification
G04BE03 - sildenafil ; Belongs to the class of drugs used in erectile dysfunction.
Presentation/Packing
Form
Zifagra FC caplet 100 mg
Packing/Price
3 × 6's
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