Angina pectoris, Hypertension
Adult: 50 mg once daily increased if necessary.
Indications and Dosage
Oral
Angina pectoris, Hypertension Adult: 50 mg once daily increased if necessary.
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Contraindications
Cardiac conduction disorders.
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Special Precautions
Elderly.
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Adverse Reactions
Abdominal pain, belching, heartburn, flushing, headache, nausea and vomiting, dizziness, lightheadedness, bradycardia, peripheral oedema, chest pain.
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Drug Interactions
Potentially Fatal: Due to its CYP3A4 and CYP2D6 inhibiting effects, serious interactions have been reported with: β-blockers, diltiazem, verapamil, digitalis glycosides, atorvastatin, cerivastatin, lovastatin, simvastatin, astemizole, cisapride, terfenadine, ciclosporin, desipramine, imipramine, tacrolimus, flecainide, propafenone.
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Action
Description: Mibefradil is a calcium channel blocker which acts principally on fast T-type calcium channels.
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MIMS Class
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